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- (R)-baclofen 69308-37-8
- (R)-baclofen 69308-37-8
(R)-baclofen 69308-37-8
产品描述 描述 (R)-baclofena， a derivative of gamma-aminobutyric acid，is commonly utilized for the treatment of spasticity.
纯度 ＞98%储存/保存方法 Store at -20℃ for one year（Powder）；Store at 2-4℃ for two weeks；Store at -20℃ for six months after dissolution.基本信息 别名 (R)-ba氯芬；STX209外观 白色粉末可溶性/溶解性 water : 4.3 mg/mL (20 mM), with gentle warming生物活性 靶点 GABAB receptorIn vitro(体外研究) Baclofen is a skeletal muscle relaxant used in the treatment of spasticity of spinal and cerebral origin. Although it is marketed as a racemic mixture, only the baclofen R-enantiomer is stereospecifically active at so called GAGAB-receptors. Researchers believe that the enantiomers of baclofen have different properties. It is claimed that the R-(−)-enantiomer is about 100 times more active than the S-(+)-enantiomer.参考文献 参考文献 研究领域 研究领域 Drug DiscoverySmall Molecule DrugLead Compound Discovery(R)-baclofen 69308-37-8温馨提示：本产品仅作科研实验使用，不支持临床等研究