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- SP600125 2mg
- SP600125 2mg
概述 描述 SP600125 is a broad-spectrum JNK inhibitor for JNK1, JNK2 and JNK3 with IC50 of 40 nM, 40 nM and 90 nM, respectively; 10-fold greater selectivity against MKK4, 25-fold greater selectivity against MKK3, MKK6, PKB, and PKCα, and 100-fold selectivity against ERK2, p38, Chk1, EGFR etc. 性能 保存方法 -20°C 分子量 220.23 化学式 C14H8N2O 分子结构式 溶解性 DMSO:44 mg/mL (199.79 mM) CAS号 129-56-6 参考文献
- 1. Bennett BL, et al. Proc Natl Acad Sci U S A, 2001, 98(24), 13681-13686.
- 2. Colombo R, et al. Cancer Res, 2010, 70(24), 10255-64.